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First Aid Kits are collections of the most important medical equipment required for quick medical assistance. Similarly, enzyme kits can provide a proficient, ready‐ and easy‐to‐use collection of biocatalysts that can be applied with high reproducibility. In this article, we illustrate how kits of oxyfunctionalisation enzymes could operate as synthetic 'First Aid' for chemists working on complex natural product total synthesis in an early‐ or late‐stage fashion, as well as in lead diversification in drug discovery processes. We reason that enzyme kits could catalyse the integration of biocatalysis into (synthetic) organic chemistry and describe how we envision their future application. [ABSTRACT FROM AUTHOR]

Biocatalysis, early-stage functionalisation, enzyme kits, late-stage functionalisation, lead diversification Cover Feature: Enzyme Kits to Facilitate the Integration of Biocatalysis into Organic Chemistry - First Aid for Synthetic Chemists (ChemCatChem 11/2022) Keywords: biocatalysis; early-stage functionalisation; enzyme kits; late-stage functionalisation; lead diversification EN biocatalysis early-stage functionalisation enzyme kits late-stage functionalisation lead diversification 1 1 1 06/10/22 20220608 NES 220608 B The Cover Feature b illustrates how enzyme kits function as proficient and readily available "First Aid" for synthetic chemists, to simplify syntheses of complex molecules complementary to conventional chemical methods. [Extracted from the article]