37 results on '"Gerona‐Navarro, Guillermo"'
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2. Abstract PO-008: Bithioether Stapled Peptides as Allosteric Inhibitors of PRC2 function
3. In silico design and molecular basis for the selectivity of Olinone toward the first over the second bromodomain of BRD4
4. Peptidomimetics Targeting Protein-Protein Interactions for Therapeutic Development
5. A Solid‐Phase Approach to Accessing Bisthioether‐Stapled Peptides Resulting in a Potent Inhibitor of PRC2 Catalytic Activity
6. A Solid‐Phase Approach to Accessing Bisthioether‐Stapled Peptides Resulting in a Potent Inhibitor of PRC2 Catalytic Activity
7. Modulating Mineralocorticoid Receptor with Non-steroidal Antagonists. New Opportunities for the Development of Potent and Selective Ligands without Off-Target Side Effects
8. Control of Embryonic Stem Cell Identity by BRD4-Dependent Transcriptional Elongation of Super-Enhancer-Associated Pluripotency Genes
9. Selective Chemical Modulation of Gene Transcription Favors Oligodendrocyte Lineage Progression
10. Cyclic amino acid linkers stabilizing key loops of brain derived neurotrophic factor
11. Solid-Phase Synthesis of a Library of Amphipatic Hydantoins. Discovery of New Hits for TRPV1 Blockade
12. A Small Molecule Binding to the Coactivator CREB-Binding Protein Blocks Apoptosis in Cardiomyocytes
13. Assembling Ligands In Situ Using Bioorthogonal Boronate Ester Synthesis
14. ChemInform Abstract: Entry to New Conformationally Constrained Amino Acids. First Synthesis of 3-Unsubstituted 4-Alkyl-4-carboxy-2-azetidinone Derivatives via an Intramolecular Nα-Cα-Cyclization Strategy.
15. ChemInform Abstract: General Approach for the Stereocontrolled Construction of the β-Lactam Ring in Amino Acid-Derived 4-Alkyl-4-carboxy-2-azetidinones.
16. Further Evidence for 2-Alkyl-2-carboxyazetidines as γ-Turn Inducers
17. Structural Basis of Site-Specific Histone Recognition by the Bromodomains of Human Coactivators PCAF and CBP/p300
18. Azetidine-Derived Amino Acids versus Proline Derivatives. Alternative Trends in Reverse Turn Induction
19. 2-Alkyl-2-carboxy-azetidines as scaffolds for the induction of γ-turns
20. From 1-Acyl-β-lactam Human Cytomegalovirus Protease Inhibitors to 1-Benzyloxycarbonylazetidines with Improved Antiviral Activity. A Straightforward Approach To Convert Covalent to Noncovalent Inhibitors
21. Ligand Discovery Using Small Molecule Microarrays
22. Synthesis and anti‐HCMV Activity of 1‐Acyl‐β‐lactams and 1‐Acylazetidines Derived from Phenylalanine.
23. Exploring Different Approaches for the Stereoselective Synthesis of Amino Acid Derived 4‐Alkyl‐4‐carboxy‐2‐azetidinones
24. Synthesis and anti-HCMV activity of 1-acyl-β-lactams and 1-acylazetidines derived from phenylalanine
25. Simple access to novel azetidine-containing conformationally restricted amino acids by chemoselective reduction of β-lactams
26. Easy Access to Orthogonally Protected α‐Alkyl Aspartic Acid and α‐Alkyl Asparagine Derivatives by Controlled Opening of β‐Lactams.
27. Memory of Chirality in the Stereoselective Synthesis of β‐Lactams: Importance of the Starting Amino Acid Derivative.
28. Memory of Chirality in the Enantioselective Synthesis of β-Lactams Derived from Amino Acids. Influence of the Reaction Conditions.
29. Memory of chirality in the stereoselective synthesis of β-lactams: importance of the starting amino acid derivative
30. Easy access to orthogonally protected α-alkyl aspartic acid and α-alkyl asparagine derivatives by controlled opening of β-lactams
31. Memory of Chirality in theEnantioselective Synthesis of β-Lactams Derived from AminoAcids. Influence of the Reaction Conditions
32. ChemInform Abstract: Amino Acid Derived 4‐Alkyl‐4‐carboxy‐2‐azetidinones. New Insights into β‐Lactam Ring Formation and N‐Deprotection.
33. General Approach for the Stereocontrolled Construction of the β-Lactam Ring in Amino Acid-Derived 4-Alkyl-4-carboxy-2-azetidinones
34. Amino Acid-derived 4-Alkyl-4-carboxy-2-azetidinones. New Insights into b-Lactam Ring Formation and N-Deprotection
35. Entry to New Conformationally Constrained Amino Acids. First Synthesis of 3-Unsubstituted 4-Alkyl-4-carboxy-2-azetidinone Derivatives via an Intramolecular Nα-Cα-Cyclization Strategy
36. ChemInform Abstract: New Conformationally Constrained Tryptophans by Nα‐Cα‐Cyclization to an Azetidin‐2‐one Core.
37. Exploring solid-phase approaches for the preparation of new -lactams from amino acids
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